Granulation Essay

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1.3 Granulation

Granulation is a common technique used to produce powders that can be compacted. In this process, the particles are enlarged via agglomeration of the particles while still maintaining the original particles integrity.

Granulation importance
• Granulation is important to prevent segregation of the particles in the powder. Segregation may be due to the different density or sizes of particles. Denser particles tend to settle at the bottom of the container while the lighter particles will tend to stay on the top.
• Granulation helps to improve the characteristics of the powder mix for compaction. Granules are often easy to compact and create stronger tablets.
• It decreases the chances for caking of partially hygroscopic materials, in case of storage as a powder. This is achieved since the moisture is adsorbed onto the surface of the granulated particles and they can still maintain their flowability due to its size(1).

There are 2 types of granulation: Wet granulation and dry granulation. As the name suggests, wet granulation requires a liquid to be used in the process of agglomeration whereas dry granulation doesn’t require any liquid. Both these processes will be discussed in detail in the upcoming sections.

1.3.1.1 Mechanism of particle agglomeration in wet Granulation
The granulation liquid (fluid) contains a solvent which must be volatile so that it can be removed by drying and be non-toxic. Typical liquids include water, ethanol and isopropanol either alone or in combination(2).The liquid solution can be either aqueous based or solvent based. Aqueous solutions have the advantage of being safer to deal with than solvents. Water also has disadvantages as a solvent since it can affect drug stability adversel...

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... than that required for making a tablet via direct compression.
• Due to the addition of water, entrapped air is decreased which reduces the dustiness as compared to dry granulation.
• Prevents the segregation of the components by forming a homogeneous powder.
• Dissolution rate of hydrophobic drugs is improved due to certain binders and solvents.

Disadvantages of wet granulation are:

• This method is expensive due to cost of time, equipment, energy and space requirements as compared to direct compression.
• Increased number of processing units increases the chance of problems such as difficulty in controlling or validation.
• Air and vapour handling equipment needs to be in place to get rid of vapour in case of solvent being a health hazard.
• Incompactibity between the components of formulation will be aggravated due to being in contact with the solvent(2).

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